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Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31b

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Protein Data Bank Japan2025-10-01 更新2026-03-21 收录
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Structure of human methionine aminopeptidase-2 complexed with spiroepoxytriazole inhibitor (+)-31b Descriptor: (4S,7R)-7-hydroxy-1-(4-methoxybenzyl)-7-methyl-4,5,6,7-tetrahydro-1H-benzotriazol-4-yl propan-2-ylcarbamate, 1,2-ETHANEDIOL, COBALT (II) ION, ... Authors: Janowski, R, Miller, A.K, Niessing, D. Deposit date: 2015-08-12 Release date: 2016-01-13 Last modified: 2025-10-01 Method: X-RAY DIFFRACTION (1.55 Å) Cite: Spiroepoxytriazoles Are Fumagillin-like Irreversible Inhibitors of MetAP2 with Potent Cellular Activity. Acs Chem.Biol., 11, 2016
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2015-08-12
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