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Protein Kinase A in complex with an Inhibitor

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Protein Kinase A in complex with an Inhibitor Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, 7-[(3S,4R)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3H-quinazolin-4-one, CAMP-DEPENDENT PROTEIN KINASE CATALYTIC SUBUNIT ALPHA, ... Authors: Alam, K.A, Engh, R.A. Deposit date: 2015-04-07 Release date: 2016-04-13 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (1.768 Å) Cite: Addressing the Glycine-Rich Loop of Protein Kinases by a Multi-Facetted Interaction Network: Inhibition of Pka and a Pkb Mimic. Chemistry, 22, 2016
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2015-04-07
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