Crystal structure of human 14-3-3 sigma in complex with TASK-3 peptide and stabilizer 16-O-Me-FC-H
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Crystal structure of human 14-3-3 sigma in complex with TASK-3 peptide and stabilizer 16-O-Me-FC-H Descriptor: (4R,5R,6R,6aS,9S,9aE,10aR)-5-hydroxy-9-(methoxymethyl)-6,10a-dimethyl-3-(propan-2-yl)-1,2,4,5,6,6a,7,8,9,10a-decahydrodicyclopenta[a,d][8]annulen-4-yl alpha-D-glucopyranoside, 14-3-3 protein sigma, MAGNESIUM ION, ... Authors: Ottmann, C, Anders, C, Schumacher, B. Deposit date: 2012-06-26 Release date: 2013-05-08 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.9 Å) Cite: A semisynthetic fusicoccane stabilizes a protein-protein interaction and enhances the expression of k(+) channels at the cell surface. Chem.Biol., 20, 2013
人类14-3-3σ(14-3-3 sigma)与TASK-3肽及稳定剂16-O-Me-FC-H结合的晶体结构 结构表征:(4R,5R,6R,6aS,9S,9aE,10aR)-5-羟基-9-(甲氧基甲基)-6,10a-二甲基-3-(异丙基)-1,2,4,5,6,6a,7,8,9,10a-十氢二环戊并[a,d][8]轮烯-4-基 α-D-吡喃葡萄糖苷、14-3-3蛋白σ亚型、镁离子(MAGNESIUM ION)等 作者:Ottmann, C、Anders, C、Schumacher, B 提交日期:2012-06-26 发布日期:2013-05-08 最后修改日期:2024-11-20 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.9埃 引用文献:一种半合成壳梭孢烷类化合物可稳定蛋白质-蛋白质相互作用并增强细胞表面钾离子通道的表达,《Chem.Biol.》,20卷,2013年



