p53 cancer mutant Y220S in complex with small-molecule stabilizer PK9323
收藏Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6si4
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p53 cancer mutant Y220S in complex with small-molecule stabilizer PK9323 Descriptor: 1-[9-ethyl-7-(1,3-thiazol-4-yl)carbazol-3-yl]-~{N}-methyl-methanamine, Cellular tumor antigen p53, GLYCEROL, ... Authors: Joerger, A.C, Kraemer, A, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2019-08-08 Release date: 2020-02-19 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Targeting Cavity-Creating p53 Cancer Mutations with Small-Molecule Stabilizers: the Y220X Paradigm. Acs Chem.Biol., 15, 2020
创建时间:
2019-08-08



