Structure of human GLP SET-domain (EHMT1) in complex with covalent inhibitor (Compound 1)
收藏Protein Data Bank Japan2024-11-06 更新2026-04-25 收录
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Structure of human GLP SET-domain (EHMT1) in complex with covalent inhibitor (Compound 1) Descriptor: Histone-lysine N-methyltransferase EHMT1, N-(6-methoxy-4-{[1-(propan-2-yl)piperidin-4-yl]amino}-7-[3-(pyrrolidin-1-yl)propoxy]quinazolin-2-yl)prop-2-enamide, N-(6-methoxy-4-{[1-(propan-2-yl)piperidin-4-yl]amino}-7-[3-(pyrrolidin-1-yl)propoxy]quinazolin-2-yl)propanamide, ... Authors: Park, K.-S, Kumar, P. Deposit date: 2021-12-15 Release date: 2022-07-06 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Discovery of the First-in-Class G9a/GLP Covalent Inhibitors. J.Med.Chem., 65, 2022
创建时间：
2021-12-15
