CLK1 bound with benzothiazole Tg003 (Cpd 2)
收藏Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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CLK1 bound with benzothiazole Tg003 (Cpd 2) Descriptor: (1~{Z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one, Dual specificity protein kinase CLK1 Authors: Schroeder, M, Chaikuad, A, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2020-04-24 Release date: 2020-07-15 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.3 Å) Cite: DFG-1 Residue Controls Inhibitor Binding Mode and Affinity, Providing a Basis for Rational Design of Kinase Inhibitor Selectivity. J.Med.Chem., 63, 2020
创建时间:
2020-04-24



