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Crystal structure of ATAD2A bromodomain complexed with 3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[(phenylsulfonyl)amino]benzoicacid

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Crystal structure of ATAD2A bromodomain complexed with 3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[(phenylsulfonyl)amino]benzoicacid Descriptor: 3-(3,5-dimethyl-1,2-oxazol-4-yl)-5-[(phenylsulfonyl)amino]benzoic acid, ATPase family AAA domain-containing protein 2, CHLORIDE ION, ... Authors: Poncet-Montange, G, Zhan, Y, Bardenhagen, J, Petrocchi, A, Leo, E, Shi, X, Lee, G, Leonard, P, Geck Do, M, Cardozo, M, Palmer, W, Andersen, J, Jones, P, Ladbury, J. Deposit date: 2014-06-23 Release date: 2014-12-24 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (1.73 Å) Cite: Observed bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2. Biochem.J., 466, 2015

ATAD2A溴结构域(bromodomain)与3-(3,5-二甲基-1,2-恶唑-4-基)-5-[(苯磺酰基)氨基]苯甲酸共晶的晶体结构 描述符:3-(3,5-二甲基-1,2-恶唑-4-基)-5-[(苯磺酰基)氨基]苯甲酸、ATP酶家族AAA结构域包含蛋白2(ATPase family AAA domain-containing protein 2)、氯离子(CHLORIDE ION)等 作者:Poncet-Montange, G、Zhan, Y、Bardenhagen, J、Petrocchi, A、Leo, E、Shi, X、Lee, G、Leonard, P、Geck Do, M、Cardozo, M、Palmer, W、Andersen, J、Jones, P、Ladbury, J 存档日期:2014-06-23 发布日期:2014-12-24 末次修改日期:2023-09-27 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.73 Å 引用文献:《溴结构域的柔性观测揭示ATAD2的组蛋白肽与小分子配体兼容构象》,Biochem.J., 466, 2015
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2014-06-23
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