PDK1 mutant bound to allosteric disulfide fragment activator JS30
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https://pdbj.org/mine/summary/3otu
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PDK1 mutant bound to allosteric disulfide fragment activator JS30 Descriptor: 3-(1H-INDOL-3-YL)-4-{1-[2-(1-METHYLPYRROLIDIN-2-YL)ETHYL]-1H-INDOL-3-YL}-1H-PYRROLE-2,5-DIONE, 3-phosphoinositide-dependent protein kinase 1, 4-[4-(naphthalen-1-ylmethyl)piperazin-1-yl]-4-oxobutane-1-thiol, ... Authors: Sadowsky, J.D, Wells, J.A. Deposit date: 2010-09-13 Release date: 2011-03-23 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (2.1013 Å) Cite: Turning a protein kinase on or off from a single allosteric site via disulfide trapping. Proc.Natl.Acad.Sci.USA, 108, 2011
创建时间:
2010-09-13



