Crystal structure of CK1 delta in complex with PK-09-129
收藏Protein Data Bank Japan2024-02-07 更新2026-04-25 收录
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Crystal structure of CK1 delta in complex with PK-09-129 Descriptor: 3-(dimethylamino)-~{N}-[4-[4-(4-fluorophenyl)-5-(1~{H}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide, Casein kinase I isoform delta, SULFATE ION Authors: Chaikuad, A, Khirsariya, P, Paruch, K, Knapp, S, Structural Genomics Consortium (SGC) Deposit date: 2022-01-10 Release date: 2023-01-18 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity. Angew.Chem.Int.Ed.Engl., 62, 2023
创建时间:
2022-01-10



