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Crystal structure of C-terminal Domain of MSK1 in complex with covalently bound pyrrolopyrimidine compound 20 (co-crystal)

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Protein Data Bank Japan2024-10-30 更新2026-04-19 收录
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Crystal structure of C-terminal Domain of MSK1 in complex with covalently bound pyrrolopyrimidine compound 20 (co-crystal) Descriptor: (5M)-5-(2,5-dichloropyrimidin-4-yl)-5H-pyrrolo[3,2-d]pyrimidine, Ribosomal protein S6 kinase alpha-5 Authors: Yano, J.K, Abendroth, J, Hall, A. Deposit date: 2022-04-14 Release date: 2022-07-06 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (3 Å) Cite: Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1. Acs Med.Chem.Lett., 13, 2022
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2022-04-14
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