Structure of cytochrome P450 EryK in complex with inhibitor ketoconazole (KC)
收藏Protein Data Bank Japan2023-12-13 更新2026-03-21 收录
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Structure of cytochrome P450 EryK in complex with inhibitor ketoconazole (KC) Descriptor: 1-ACETYL-4-(4-{[(2S,4R)-2-(2,4-DICHLOROPHENYL)-2-(1H-IMIDAZOL-1-YLMETHYL)-1,3-DIOXOLAN-4-YL]METHOXY}PHENYL)PIPERAZINE, CYTOCHROME P450 113A1, PROTOPORPHYRIN IX CONTAINING FE, ... Authors: Savino, C, Sciara, G, Miele, A.E, Kendrew, S.G, Vallone, B. Deposit date: 2008-04-15 Release date: 2009-07-14 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Azole Drugs Trap Cytochrome P450 Eryk in Alternative Conformational States. Biochemistry, 49, 2010
创建时间:
2008-04-15



