Selective PI3K beta inhibitor bound to PI3K delta
收藏Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6dgt
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Selective PI3K beta inhibitor bound to PI3K delta Descriptor: 4-[1-(5,8-difluoroquinolin-4-yl)-2-methyl-4-(4H-1,2,4-triazol-3-yl)-1H-benzimidazol-6-yl]-3-fluoropyridin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform Authors: Somoza, J, Villasenor, A, McGrath, M. Deposit date: 2018-05-18 Release date: 2018-08-01 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.601 Å) Cite: Atropisomerism by Design: Discovery of a Selective and Stable Phosphoinositide 3-Kinase (PI3K) beta Inhibitor. J. Med. Chem., 61, 2018
创建时间:
2018-05-18



