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HIV-1 protease-inhibitor complex

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Protein Data Bank Japan2024-02-14 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2bpw
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HIV-1 protease-inhibitor complex Descriptor: 1-[2-HYDROXY-4-(2-HYDROXY-5-METHYL-CYCLOPENTYLCARBAMOYL)5-PHENYL-PENTYL]-4-(3-PYRIDIN-3-YL-PROPIONYL)-PIPERAZINE-2-CARB OXYLIC ACID TERT-BUTYLAMIDE, HIV-1 PROTEASE Authors: Munshi, S, Chen, Z. Deposit date: 1998-01-22 Release date: 1999-02-23 Last modified: 2024-02-14 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Rapid X-ray diffraction analysis of HIV-1 protease-inhibitor complexes: inhibitor exchange in single crystals of the bound enzyme. Acta Crystallogr.,Sect.D, 54, 1998

HIV-1蛋白酶-抑制剂复合物(HIV-1 protease-inhibitor complex) 描述符:1-[2-羟基-4-(2-羟基-5-甲基-环戊基甲酰基)-5-苯基-戊基]-4-(3-吡啶-3-基-丙酰基)-哌嗪-2-羧酸叔丁酰胺(1-[2-HYDROXY-4-(2-HYDROXY-5-METHYL-CYCLOPENTYLCARBAMOYL)5-PHENYL-PENTYL]-4-(3-PYRIDIN-3-YL-PROPIONYL)-PIPERAZINE-2-CARBOXYLIC ACID TERT-BUTYLAMIDE) 作者:Munshi, S、Chen, Z. 存入日期:1998-01-22 发布日期:1999-02-23 最后修改日期:2024-02-14 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率2.8埃(2.8 Å) 引用:《HIV-1蛋白酶-抑制剂复合物的快速X射线衍射分析:结合酶单晶体中的抑制剂交换》,《Acta Crystallogr., Sect. D》(《晶体学报D辑》),54卷,1998年
创建时间:
1998-01-22
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