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Studies Towards a Reversible EGFR C797S Triple Mutant Inhibitor Series

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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Studies Towards a Reversible EGFR C797S Triple Mutant Inhibitor Series Descriptor: 5-chloranyl-~{N}2-[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-5-(1-methylpyrazol-4-yl)phenyl]-~{N}4-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamine, Epidermal growth factor receptor Authors: Hargreaves, D. Deposit date: 2020-09-17 Release date: 2021-06-02 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (2.65 Å) Cite: Abstract 4451: Evaluation of the therapeutic potential of phosphine oxide pyrazole inhibitors in tumors harboring EGFR C797S mutation Cancer Res., 79, 2019
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2020-09-17
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