five

SRPK1 in complex with Alectinib

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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SRPK1 in complex with Alectinib Descriptor: 1,2-ETHANEDIOL, 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5H-benzo[b]carbazole-3-carbonitrile, serine-arginine (SR) protein kinase 1 Authors: Zeng, C, Ngo, J.C.K. Deposit date: 2017-06-26 Release date: 2018-03-14 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (2.32 Å) Cite: SRPKIN-1: A Covalent SRPK1/2 Inhibitor that Potently Converts VEGF from Pro-angiogenic to Anti-angiogenic Isoform Cell Chem Biol, 25, 2018
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2017-06-26
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