Crystal Structure of PI3Kalpha in complex with fragment 10
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Crystal Structure of PI3Kalpha in complex with fragment 10 Descriptor: 2-(trifluoromethyl)-1H-benzimidazol-5-amine, Phosphatidylinositol 3-kinase regulatory subunit alpha, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform Authors: Gabelli, S.B, Vogelstein, B, Miller, M.S, Amzel, L.M. Deposit date: 2016-08-09 Release date: 2017-02-15 Last modified: 2024-10-09 Method: X-RAY DIFFRACTION (3.35 Å) Cite: Identification of allosteric binding sites for PI3K alpha oncogenic mutant specific inhibitor design. Bioorg. Med. Chem., 25, 2017
创建时间:
2016-08-09



