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Human MTHFD2 in complex with compound 21 and 15

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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Human MTHFD2 in complex with compound 21 and 15 Descriptor: (2S)-2-[[4-[(4-azanyl-6-oxidanyl-pyrimidin-5-yl)carbamoylamino]phenyl]carbonylamino]pentanedioic acid, (2S)-2-[[4-[[1-[(3,4-dichlorophenyl)methyl]-3,7-dimethyl-2,6-bis(oxidanylidene)purin-8-yl]amino]phenyl]carbonylamino]pentanedioic acid, Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, ... Authors: Lee, L.C, Peng, Y.H, Wu, S.Y. Deposit date: 2021-03-30 Release date: 2021-08-11 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.13 Å) Cite: Xanthine Derivatives Reveal an Allosteric Binding Site in Methylenetetrahydrofolate Dehydrogenase 2 (MTHFD2). J.Med.Chem., 64, 2021
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2021-03-30
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