five

TTK kinase domain in complex with BAY 1161909

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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TTK kinase domain in complex with BAY 1161909 Descriptor: (2~{R})-2-(4-fluorophenyl)-~{N}-[4-[2-[(2-methoxy-4-methylsulfonyl-phenyl)amino]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamide, Dual specificity protein kinase TTK Authors: Uitdehaag, J, Willemsen-Seegers, N, de Man, J, Buijsman, R.C, Zaman, G.J.R. Deposit date: 2017-02-27 Release date: 2017-05-31 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity. J. Mol. Biol., 429, 2017
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2017-02-27
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