five

N-terminal bromodomain of BRD4 in complex with OTX-015

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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N-terminal bromodomain of BRD4 in complex with OTX-015 Descriptor: 2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-(4-hydroxyphenyl)acetamide, Bromodomain-containing protein 4 Authors: Zhang, Y. Deposit date: 2017-07-28 Release date: 2018-08-01 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.27 Å) Cite: BRD4 Profiling Identifies Critical Chronic Lymphocytic Leukemia Oncogenic Circuits and Reveals Sensitivity to PLX51107, a Novel Structurally Distinct BET Inhibitor. Cancer Discov, 8, 2018
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2017-07-28
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