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Encequidar-bound human P-glycoprotein in complex with UIC2-Fab

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Protein Data Bank Japan2025-07-02 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7o9w
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Encequidar-bound human P-glycoprotein in complex with UIC2-Fab Descriptor: Multidrug resistance protein 1, UIC2 Fab-fragment heavy chain, UIC2 Fab-fragment light chain, ... Authors: Nosol, K, Locher, K.P. Deposit date: 2021-04-17 Release date: 2022-01-12 Last modified: 2025-07-02 Method: ELECTRON MICROSCOPY (3.5 Å) Cite: Discovery and Characterization of Potent Dual P-Glycoprotein and CYP3A4 Inhibitors: Design, Synthesis, Cryo-EM Analysis, and Biological Evaluations. J.Med.Chem., 65, 2022
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2021-04-17
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