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CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE PEPTIDE SUBSTRATE TKCVFM AND AN ANALOG OF FARNESYL DIPHOSPHATE

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Protein Data Bank Japan2023-08-16 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE PEPTIDE SUBSTRATE TKCVFM AND AN ANALOG OF FARNESYL DIPHOSPHATE Descriptor: ACETIC ACID, PROTEIN FARNESYLTRANSFERASE, ALPHA SUBUNIT, ... Authors: Long, S.B, Casey, P.J, Beese, L.S. Deposit date: 2001-06-11 Release date: 2001-11-02 Last modified: 2023-08-16 Method: X-RAY DIFFRACTION (2.2 Å) Cite: The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98, 2001
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2001-06-11
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