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Crystal structure of HUMAN WEE1 KINASE domain in complex with Bosutinib-isomer

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5vc4
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Crystal structure of HUMAN WEE1 KINASE domain in complex with Bosutinib-isomer Descriptor: 4-[(3,5-DICHLORO-4-METHOXYPHENYL)AMINO]-6-METHOXY-7-[3-(4-METHYLPIPERAZIN-1-YL)PROPOXY]QUINOLINE-3-CARBONITRILE, PHOSPHATE ION, Wee1-like protein kinase Authors: Zhu, J.-Y, Schonbrunn, E. Deposit date: 2017-03-30 Release date: 2017-08-23 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors. J. Med. Chem., 60, 2017
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2017-03-30
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