Crystal structure of RPE65 in complex with MB-008 and palmitate
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Crystal structure of RPE65 in complex with MB-008 and palmitate Descriptor: (3S)-3-({3-[(1R)-3-amino-1-hydroxypropyl]phenoxy}methyl)hexan-1-ol, FE (II) ION, PALMITIC ACID, ... Authors: Kiser, P.D, Palczewski, K. Deposit date: 2017-01-24 Release date: 2017-05-17 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Rational Tuning of Visual Cycle Modulator Pharmacodynamics. J. Pharmacol. Exp. Ther., 362, 2017
结合MB-008与棕榈酸的RPE65晶体结构 配体描述:(3S)-3-({3-[(1R)-3-氨基-1-羟丙基]苯氧基}甲基)己-1-醇、二价铁离子(Fe(II) ION)、棕榈酸(PALMITIC ACID)…… 作者:Kiser, P.D.、Palczewski, K. 沉积日期:2017-01-24 发布日期:2017-05-17 最后修改日期:2023-10-04 实验方法:X射线衍射(X-RAY DIFFRACTION,分辨率2.1埃(Å)) 引用文献:《视觉循环调节剂药效学的理性优化》,载于《药理学与实验治疗学杂志》(J. Pharmacol. Exp. Ther.),第362卷,2017年
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2017-01-24



