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Human JNK2 bound to covalent inhibitor YL2056

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Protein Data Bank Japan2024-11-13 更新2026-04-25 收录
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资源简介:
Human JNK2 bound to covalent inhibitor YL2056 Descriptor: 4-(dimethylamino)-N-{4-[(3S)-3-({4-[(8R)-2-phenylpyrazolo[1,5-a]pyridin-3-yl]pyrimidin-2-yl}amino)pyrrolidine-1-carbonyl]phenyl}butanamide, Mitogen-activated protein kinase 9 Authors: Li, L, Gurbani, D, Westover, K.D. Deposit date: 2022-09-23 Release date: 2023-06-28 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.072 Å) Cite: Development of a Covalent Inhibitor of c-Jun N-Terminal Protein Kinase (JNK) 2/3 with Selectivity over JNK1. J.Med.Chem., 66, 2023
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2022-09-23
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