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Structure of the 50S ribosomal subunit from Methicillin Resistant Staphylococcus aureus in complex with the oxazolidinone antibiotic LZD-5

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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Structure of the 50S ribosomal subunit from Methicillin Resistant Staphylococcus aureus in complex with the oxazolidinone antibiotic LZD-5 Descriptor: 2,2-dichloro-N-({(5S)-3-[3-fluoro-4-(morpholin-4-yl)phenyl]-2-oxo-1,3-oxazolidin-5-yl}methyl)acetamide, 23S rRNA, 50S ribosomal protein L13, ... Authors: Belousoff, M.J, Venugopal, H, Bamert, R.S, Lithgow, T. Deposit date: 2018-05-10 Release date: 2019-03-20 Last modified: 2024-10-16 Method: ELECTRON MICROSCOPY (3.1 Å) Cite: cryoEM-Guided Development of Antibiotics for Drug-Resistant Bacteria. ChemMedChem, 14, 2019

耐甲氧西林金黄色葡萄球菌(Methicillin Resistant Staphylococcus aureus)来源的50S核糖体亚基(50S ribosomal subunit)与恶唑烷酮类抗生素(oxazolidinone antibiotic)LZD-5形成复合物的结构 结构描述:2,2-二氯-N-({(5S)-3-[3-氟-4-(4-吗啉基)苯基]-2-氧代-1,3-恶唑烷-5-基}甲基)乙酰胺、23S核糖体RNA(23S rRNA)、50S核糖体蛋白L13等 作者:Belousoff, M.J.、Venugopal, H.、Bamert, R.S.、Lithgow, T. 提交日期:2018-05-10 发布日期:2019-03-20 最后修改日期:2024-10-16 实验方法:电子显微镜(分辨率3.1 Å) 引用文献:《冷冻电镜指导耐药细菌用抗生素开发》,ChemMedChem,第14卷,2019年
创建时间:
2018-05-10
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