five

Crystal structure of VIM-2 in complex with triazole-based inhibitor OP24

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Crystal structure of VIM-2 in complex with triazole-based inhibitor OP24 Descriptor: 5-(4-chloranyl-1,5-dimethyl-pyrazol-3-yl)-4-ethyl-1,2,4-triazole-3-thiol, FORMIC ACID, Vim-1, ... Authors: Maso, L, Spirakis, F, Santucci, M, Simon, C, Docquier, J.D, Cruciani, G, Costi, M.P, Tondi, D, Cendron, L. Deposit date: 2019-11-15 Release date: 2020-10-14 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (1.6 Å) Cite: Virtual screening identifies broad-spectrum beta-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases. Sci Rep, 10, 2020
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2019-11-15
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