Crystal Structure Analysis of the 1,2,3-tricarboxylate benzoic acid bound to sp-ASADH-2'5'-ADP complex
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Crystal Structure Analysis of the 1,2,3-tricarboxylate benzoic acid bound to sp-ASADH-2'5'-ADP complex Descriptor: 1,2-ETHANEDIOL, ACETATE ION, ADENOSINE-2'-5'-DIPHOSPHATE, ... Authors: Pavlovsky, A.G, Viola, R.E. Deposit date: 2014-08-18 Release date: 2014-12-10 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.91 Å) Cite: A cautionary tale of structure-guided inhibitor development against an essential enzyme in the aspartate-biosynthetic pathway. Acta Crystallogr.,Sect.D, 70, 2014
结合sp-ASADH-2'5'-二磷酸腺苷复合物的1,2,3-三羧基苯甲酸的晶体结构分析
配体描述:1,2-乙二醇、乙酸根离子、腺苷-2',5'-二磷酸(ADENOSINE-2'-5'-DIPHOSPHATE)……
作者:帕夫洛夫斯基(Pavlovsky, A.G)、维奥拉(Viola, R.E.)
存档日期:2014-08-18
发布日期:2014-12-10
最后修改日期:2023-09-20
实验方法:X射线衍射(分辨率1.91埃)
引用文献:《天冬氨酸生物合成途径中关键酶的结构导向抑制剂开发的警示案例》,《Acta Crystallogr.,Sect.D》,第70卷,2014年
创建时间:
2014-08-18



