Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design
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Differential Binding Of Inhibitors To Active And Inactive Cdk2 Provides Insights For Drug Design Descriptor: CELL DIVISION PROTEIN KINASE 2, CYCLIN A2, HYDROXY(OXO)(3-{[(2Z)-4-[3-(1H-1,2,4-TRIAZOL-1-YLMETHYL)PHENYL]PYRIMIDIN-2(5H)-YLIDENE]AMINO}PHENYL)AMMONIUM Authors: Kontopidis, G, Mcinnes, C, Pandalaneni, S.R, Mcnae, I, Gibson, D, Mezna, M, Thomas, M, Wood, G, Wang, S, Walkinshaw, M.D, Fischer, P.M. Deposit date: 2005-11-03 Release date: 2006-03-01 Last modified: 2023-12-13 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Differential Binding of Inhibitors to Active and Inactive Cdk2 Provides Insights for Drug Design. Chem.Biol., 13, 2006
抑制剂与活性及非活性Cdk2的差异化结合为药物设计提供启示 描述符:细胞分裂蛋白激酶2(CELL DIVISION PROTEIN KINASE 2)、细胞周期蛋白A2(CYCLIN A2)、HYDROXY(OXO)(3-{[(2Z)-4-[3-(1H-1,2,4-TRIAZOL-1-YLMETHYL)PHENYL]PYRIMIDIN-2(5H)-YLIDENE]AMINO}PHENYL)AMMONIUM 作者:Kontopidis G、Mcinnes C、Pandalaneni S.R、Mcnae I、Gibson D、Mezna M、Thomas M、Wood G、Wang S、Walkinshaw M.D、Fischer P.M. 提交日期:2005年11月3日 发布日期:2006年3月1日 最后修改日期:2023年12月13日 实验方法:X射线衍射(2.9埃) 引用文献:Differential Binding of Inhibitors to Active and Inactive Cdk2 Provides Insights for Drug Design. Chem.Biol., 13, 2006



