five

Crystal structure of BRD4-BD1 bound with hjp126

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Protein Data Bank Japan2024-03-27 更新2026-03-21 收录
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Crystal structure of BRD4-BD1 bound with hjp126 Descriptor: (3~{R})-4-cyclopentyl-~{N}-(2,4-dimethylphenyl)-1,3-dimethyl-2-oxidanylidene-3~{H}-quinoxaline-6-carboxamide, Bromodomain-containing protein 4 Authors: Xiong, B, Hu, J, Li, Y, Cao, D. Deposit date: 2017-10-31 Release date: 2018-11-07 Last modified: 2024-03-27 Method: X-RAY DIFFRACTION (1.451 Å) Cite: Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups. Eur.J.Med.Chem., 150, 2018
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2017-10-31
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