Pyrazole Carboxylic Acid Inhibitors of KEAP1:NRF2 interaction
收藏Protein Data Bank Japan2024-06-19 更新2026-04-25 收录
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Pyrazole Carboxylic Acid Inhibitors of KEAP1:NRF2 interaction Descriptor: 1-[6-(3-propan-2-yloxyphenyl)pyridin-2-yl]-5-(trifluoromethyl)pyrazole-4-carboxylic acid, CHLORIDE ION, DIMETHYL SULFOXIDE, ... Authors: Davies, T.G. Deposit date: 2021-07-14 Release date: 2021-11-17 Last modified: 2024-06-19 Method: X-RAY DIFFRACTION (1.886 Å) Cite: Fragment-Guided Discovery of Pyrazole Carboxylic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2 Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction. J.Med.Chem., 64, 2021
创建时间:
2021-07-14



