Human kallikrein-related peptidase 2 in complex with PPACK
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Human kallikrein-related peptidase 2 in complex with PPACK Descriptor: D-phenylalanyl-N-[(2S,3S)-6-{[amino(iminio)methyl]amino}-1-chloro-2-hydroxyhexan-3-yl]-L-prolinamide, Kallikrein-2 Authors: Skala, W, Brandstetter, H, Magdolen, V, Goettig, P. Deposit date: 2013-10-31 Release date: 2014-10-29 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Structure-function analyses of human kallikrein-related peptidase 2 establish the 99-loop as master regulator of activity J.Biol.Chem., 289, 2014
与PPACK结合的人激肽释放酶相关肽酶2(Human kallikrein-related peptidase 2)复合物
描述物:D-苯丙氨酰-N-[(2S,3S)-6-{[氨基(亚氨基)甲基]氨基}-1-氯-2-羟基己-3-基]-L-脯氨酰胺,激肽释放酶-2
作者:Skala W、Brandstetter H、Magdolen V、Goettig P
提交日期:2013-10-31
发布日期:2014-10-29
最后更新日期:2024-10-30
实验方法:X射线衍射(分辨率1.9 Å)
引用文献:人激肽释放酶相关肽酶2的结构功能分析确立99环为活性核心调控因子,《Journal of Biological Chemistry》,289卷,2014年
创建时间:
2013-10-31



