TEAD2 bound to Compound 1
收藏Protein Data Bank Japan2023-10-25 更新2026-04-19 收录
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TEAD2 bound to Compound 1 Descriptor: Transcriptional enhancer factor TEF-4, ethyl (8S)-7-oxo-5-[4-(trifluoromethyl)phenyl]-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxylate Authors: Noland, C.L, Fong, R. Deposit date: 2022-02-14 Release date: 2023-05-03 Last modified: 2023-10-25 Method: X-RAY DIFFRACTION (1.88 Å) Cite: Novel mechanism of YAP-TEAD inhibition results in targeted chromatin remodeling and reveals an expanded Hippo dependent landscape in cancers To Be Published
创建时间:
2022-02-14



