five

Human Brd2(BD2) mutant in complex with AL-Am1

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Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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Human Brd2(BD2) mutant in complex with AL-Am1 Descriptor: (2~{R})-2-[(4~{S})-6-(4-chlorophenyl)-8-methoxy-1-methyl-4~{H}-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-~{N}-ethyl-pent-4-enamide, Bromodomain-containing protein 2 Authors: Chan, K.-H, Runcie, A.C, Ciulli, A. Deposit date: 2017-05-23 Release date: 2018-02-14 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition. Chem Sci, 9, 2018
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2017-05-23
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