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17beta-hydroxysteroid dehydrogenase type1 complexed with E2B

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Protein Data Bank Japan2024-02-21 更新2026-03-21 收录
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https://pdbj.org/mine/summary/3hb4
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资源简介:
17beta-hydroxysteroid dehydrogenase type1 complexed with E2B Descriptor: 3-{[(9beta,14beta,16alpha,17alpha)-3,17-dihydroxyestra-1,3,5(10)-trien-16-yl]methyl}benzamide, Estradiol 17-beta-dehydrogenase 1 Authors: Mazumdar, M, Fournier, D, Zhu, D.-W, Cadot, C, Poirier, D, Lin, S.-X. Deposit date: 2009-05-04 Release date: 2009-12-15 Last modified: 2024-02-21 Method: X-RAY DIFFRACTION (2.21 Å) Cite: Binary and ternary crystal structure analyses of a novel inhibitor with 17beta-HSD type 1: a lead compound for breast cancer therapy. Biochem.J., 424, 2009
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2009-05-04
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