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Human wtSTING in complex with 2',2'-difluoro-3',3'-c-di-GMP

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Protein Data Bank Japan2024-01-24 更新2026-03-21 收录
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Human wtSTING in complex with 2',2'-difluoro-3',3'-c-di-GMP Descriptor: 2-azanyl-9-[(1~{R},6~{R},8~{R},9~{R},10~{R},15~{R},17~{R},18~{R})-17-(2-azanyl-6-oxidanylidene-1~{H}-purin-9-yl)-9,18-bis(fluoranyl)-3,12-bis(oxidanyl)-3,12-bis(oxidanylidene)-2,4,7,11,13,16-hexaoxa-3$l^{5},12$l^{5}-diphosphatricyclo[13.3.0.0^{6,10}]octadecan-8-yl]-1~{H}-purin-6-one, Stimulator of interferon protein Authors: Boura, E, Smola, M. Deposit date: 2020-03-20 Release date: 2021-03-31 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.801 Å) Cite: Ligand Strain and Its Conformational Complexity Is a Major Factor in the Binding of Cyclic Dinucleotides to STING Protein. Angew.Chem.Int.Ed.Engl., 60, 2021
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2020-03-20
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