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Crystal Structure of TrkA kinase with ligand

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Protein Data Bank Japan2024-11-13 更新2026-03-21 收录
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Crystal Structure of TrkA kinase with ligand Descriptor: 1-[(3S,4R)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea, 2,3-DIHYDROXY-1,4-DITHIOBUTANE, High affinity nerve growth factor receptor, ... Authors: Noritaka, F. Deposit date: 2016-10-26 Release date: 2017-02-22 Last modified: 2024-11-13 Method: X-RAY DIFFRACTION (2.1 Å) Cite: The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity Bioorg. Med. Chem. Lett., 27, 2017
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2016-10-26
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