five

Complex of SETD8 with MS453

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Complex of SETD8 with MS453 Descriptor: 1,2-ETHANEDIOL, N-(3-{[6,7-dimethoxy-2-(pyrrolidin-1-yl)quinazolin-4-yl]amino}propyl)propanamide, N-lysine methyltransferase KMT5A, ... Authors: Yu, W, Tempel, W, Babault, N, Ma, A, Butler, K.V, Jin, J, Arrowsmith, C.H, Bountra, C, Edwards, A.M, Brown, P.J, Structural Genomics Consortium (SGC) Deposit date: 2016-09-29 Release date: 2016-11-09 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Structure-Based Design of a Covalent Inhibitor of the SET Domain-Containing Protein 8 (SETD8) Lysine Methyltransferase. J. Med. Chem., 59, 2016
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2016-09-29
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