Crystal structure of 3-oxoacyl-(acyl-carrier-protein) reductase (FabG) from Pseudomonas aeruginosa in complex with 6-(4-(2-chloroanilino)- 1H-quinazolin-2-ylidene)cyclohexa-2, 4-dien-1-one at 2.3A resolution
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Crystal structure of 3-oxoacyl-(acyl-carrier-protein) reductase (FabG) from Pseudomonas aeruginosa in complex with 6-(4-(2-chloroanilino)- 1H-quinazolin-2-ylidene)cyclohexa-2, 4-dien-1-one at 2.3A resolution Descriptor: 3-OXOACYL-[ACYL-CARRIER-PROTEIN] REDUCTASE FABG, 6-[4-(2-chloroanilino)-1H-quinazolin-2-ylidene]cyclohexa-2,4-dien-1-one Authors: Cukier, C.D, Schnell, R, Lindqvist, Y, Schneider, G. Deposit date: 2013-05-17 Release date: 2013-09-18 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Discovery of an Allosteric Inhibitor Binding Site in 3-Oxo-Acyl-Acp Reductase from Pseudomonas Aeruginosa Acs Chem.Biol., 8, 2013
铜绿假单胞菌(Pseudomonas aeruginosa)来源的3-氧酰基-[酰基载体蛋白(acyl-carrier-protein)]还原酶(FabG)与6-(4-(2-氯苯胺基)-1H-喹唑啉-2-亚基)环己-2,4-二烯-1-酮复合物的晶体结构,分辨率为2.3埃(Å)。
描述符:3-氧酰基-[酰基载体蛋白]还原酶FabG、6-[4-(2-氯苯胺基)-1H-喹唑啉-2-亚基]环己-2,4-二烯-1-酮
作者:Cukier C.D.、Schnell R.、Lindqvist Y.、Schneider G.
提交日期:2013-05-17
发布日期:2013-09-18
最后修改日期:2023-12-20
实验方法:X射线衍射(2.3 Å)
引用:《铜绿假单胞菌3-氧酰基-酰基载体蛋白还原酶变构抑制剂结合位点的发现》,《ACS化学生物学》(Acs Chem.Biol.),第8卷,2013年
创建时间:
2013-05-17



