five

Fragment-based inhibitors of Lipoprotein associated Phospholipase A2

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Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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Fragment-based inhibitors of Lipoprotein associated Phospholipase A2 Descriptor: 5-[2-(4,4-dimethyl-2-oxidanylidene-pyrrolidin-1-yl)ethoxy]-2-fluoranyl-benzenecarbonitrile, CHLORIDE ION, Platelet-activating factor acetylhydrolase Authors: Woolford, A, Day, P. Deposit date: 2016-09-29 Release date: 2016-12-21 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.07 Å) Cite: Fragment-Based Approach to the Development of an Orally Bioavailable Lactam Inhibitor of Lipoprotein-Associated Phospholipase A2 (Lp-PLA2). J. Med. Chem., 59, 2016
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2016-09-29
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