Human Deoxyhypusine Synthase Fragment Screening Campaign - ligand VT00193
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Human Deoxyhypusine Synthase Fragment Screening Campaign - ligand VT00193 Descriptor: (4R)-2-METHYLPENTANE-2,4-DIOL, 4-methylsulfonylmorpholine, Deoxyhypusine synthase, ... Authors: Wilk, P, Wator-Wilk, E, Krojer, T, Grudnik, P. Deposit date: 2025-02-15 Release date: 2026-01-21 Last modified: 2026-02-18 Method: X-RAY DIFFRACTION (1.39 Å) Cite: Crystallographic fragment screening supports tool compound discovery and reveals conformational flexibility in human deoxyhypusine synthase. Commun Chem, 9, 2026
人源脱氧羟腐胺赖氨酸合酶(Deoxyhypusine synthase)片段筛选项目——配体VT00193
描述符:(4R)-2-甲基戊烷-2,4-二醇、4-甲磺酰基吗啉、脱氧羟腐胺赖氨酸合酶……
作者:威尔克(Wilk, P)、瓦托尔-威尔克(Wator-Wilk, E)、克罗耶(Krojer, T)、格鲁德尼克(Grudnik, P)
入库日期:2025-02-15
发布日期:2026-01-21
最后修改日期:2026-02-18
实验方法:X射线衍射(1.39 Å)
引用文献:晶体片段筛选助力工具化合物发现并揭示人源脱氧羟腐胺赖氨酸合酶的构象灵活性,《通讯化学(Commun Chem)》,第9卷,2026年
创建时间:
2025-02-15



