Crsytal structure of Acinetobacter baumannii FabG inhibitor complex at 2.35 A resolution
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Crsytal structure of Acinetobacter baumannii FabG inhibitor complex at 2.35 A resolution Descriptor: 3-oxoacyl-(Acyl-carrier-protein) reductase, ethyl 6-bromanyl-2-[(dimethylamino)methyl]-5-oxidanyl-1-phenyl-indole-3-carboxylate Authors: Rudraraju, R, Schnell, R, Schneider, G. Deposit date: 2019-10-17 Release date: 2020-11-18 Last modified: 2024-01-24 Method: X-RAY DIFFRACTION (2.35 Å) Cite: A FabG inhibitor targeting an allosteric binding site inhibits several orthologs from Gram-negative ESKAPE pathogens. Bioorg.Med.Chem., 30, 2020
鲍曼不动杆菌FabG抑制剂复合物的晶体结构,分辨率2.35埃
描述符:3-氧酰基-(酰基载体蛋白)还原酶,6-溴-2-[(二甲氨基)甲基]-5-羟基-1-苯基吲哚-3-羧酸乙酯
作者:Rudraraju R、Schnell R、Schneider G
存档日期:2019-10-17
发布日期:2020-11-18
最后修改日期:2024-01-24
实验方法:X射线衍射(2.35埃)
引用文献:《靶向变构结合位点的FabG抑制剂可抑制革兰氏阴性ESKAPE病原菌的多种同源物》,《Bioorg.Med.Chem.》,2020年,第30卷
创建时间:
2019-10-17



