Crystal structure of 5beta-reductase (AKR1D1) E120H mutant in complex with NADP+ and 5beta-dihydrotestosterone
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Crystal structure of 5beta-reductase (AKR1D1) E120H mutant in complex with NADP+ and 5beta-dihydrotestosterone Descriptor: 3-oxo-5-beta-steroid 4-dehydrogenase, 5-beta-DIHYDROTESTOSTERONE, CHLORIDE ION, ... Authors: Chen, M, Christianson, D.W, Penning, T.M. Deposit date: 2011-12-07 Release date: 2012-03-21 Last modified: 2023-09-13 Method: X-RAY DIFFRACTION (1.832 Å) Cite: Conversion of Human Steroid 5beta-Reductase (AKR1D1) into 3β-Hydroxysteroid Dehydrogenase by Single Point Mutation E120H: EXAMPLE OF PERFECT ENZYME ENGINEERING. J.Biol.Chem., 287, 2012
与烟酰胺腺嘌呤二核苷酸磷酸(NADP+)和5β-二氢睾酮结合的5β-还原酶(AKR1D1)E120H突变体的晶体结构。描述符:3-氧代-5β-类固醇4-脱氢酶、5β-二氢睾酮、氯离子……。作者:Chen, M.、Christianson, D.W.、Penning, T.M.。提交日期:2011-12-07。发布日期:2012-03-21。最后修改时间:2023-09-13。实验方法:X射线衍射(分辨率1.832埃)。引用文献:《通过单点突变E120H将人类固醇5β-还原酶(AKR1D1)改造为3β-羟基类固醇脱氢酶:完美酶工程的范例》,《生物化学杂志》,287卷,2012年。
创建时间:
2011-12-07



