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Crystal Structure of COMT in complex with [3-(2,4-dimethyl-1,3-thiazol-5-yl)-1H-pyrazol-5-yl]-(4-phenylpiperazin-1-yl)methanone

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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Crystal Structure of COMT in complex with [3-(2,4-dimethyl-1,3-thiazol-5-yl)-1H-pyrazol-5-yl]-(4-phenylpiperazin-1-yl)methanone Descriptor: 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, CHLORIDE ION, Catechol O-methyltransferase, ... Authors: Ehler, A, Lerner, C, Rudolph, M.G. Deposit date: 2016-08-18 Release date: 2016-08-31 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Crystal Structure of COMT in complex with [3-(2,4-dimethyl-1,3-thiazol-5-yl)-1H-pyrazol-5-yl]-(4-phenylpiperazin-1-yl)methanone To be published

与[3-(2,4-二甲基-1,3-噻唑-5-基)-1H-吡唑-5-基]-(4-苯基哌嗪-1-基)甲酮结合的儿茶酚O-甲基转移酶(Catechol O-methyltransferase, COMT)复合物晶体结构 描述物:2-[N-环己基氨基]乙烷磺酸、氯离子、儿茶酚O-甲基转移酶等 作者:Ehler A、Lerner C、Rudolph M.G. 提交日期:2016-08-18 发布日期:2016-08-31 最后修改日期:2024-05-01 实验方法:X射线衍射(分辨率2.3 Å) 引用信息:与[3-(2,4-二甲基-1,3-噻唑-5-基)-1H-吡唑-5-基]-(4-苯基哌嗪-1-基)甲酮结合的COMT晶体结构 待发表
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2016-08-18
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