CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c12c([nH]cn1)ncnc2N(C)C3CCCCC3, micromolar IC50=3.41927
收藏Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF HUMAN PHOSPHODIESTERASE 10 IN COMPLEX WITH c12c([nH]cn1)ncnc2N(C)C3CCCCC3, micromolar IC50=3.41927 Descriptor: MAGNESIUM ION, N-cyclohexyl-N-methyl-7H-purin-6-amine, ZINC ION, ... Authors: Joseph, C, Benz, J, Flohr, A, Maurer, M, Rudolph, M.G. Deposit date: 2022-02-01 Release date: 2022-10-12 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.35 Å) Cite: Crystal Structure of a human phosphodiesterase 10 complex To be published
人源磷酸二酯酶10与c12c([nH]cn1)ncnc2N(C)C3CCCCC3复合物的晶体结构,微摩尔级半数抑制浓度(IC50)为3.41927。描述项:镁离子、N-环己基-N-甲基-7H-嘌呤-6-胺、锌离子……。作者:Joseph, C、Benz, J、Flohr, A、Maurer, M、Rudolph, M.G.。提交日期:2022-02-01,发布日期:2022-10-12,最后修改日期:2024-10-16。实验方法:X射线衍射(分辨率2.35 Å)。引用文献:《人源磷酸二酯酶10复合物的晶体结构》,待发表。
创建时间:
2022-02-01



