Structure of cyclophilin A in complex with 4-chloropyrimidin-5-amine
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Structure of cyclophilin A in complex with 4-chloropyrimidin-5-amine Descriptor: 4-chloranylpyrimidin-5-amine, Peptidyl-prolyl cis-trans isomerase A Authors: Georgiou, C, Mcnae, I.W, Ioannidis, H, Julien, M, Walkinshaw, M.D. Deposit date: 2017-04-13 Release date: 2017-07-12 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Pushing the Limits of Detection of Weak Binding Using Fragment-Based Drug Discovery: Identification of New Cyclophilin Binders. J. Mol. Biol., 429, 2017
亲环素A(cyclophilin A)与4-氯嘧啶-5-胺的复合物结构 描述物:4-氯嘧啶-5-胺,肽基脯氨酰顺反异构酶A(Peptidyl-prolyl cis-trans isomerase A) 作者:C. 乔治乌、I.W. 麦克内伊、H. 约安尼季斯、M. 朱利安、M.D. 沃金肖 提交日期:2017-04-13 发布日期:2017-07-12 最后修改日期:2024-01-17 实验方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.45埃(Å) 引用文献:《基于片段的药物发现中弱结合检测的极限突破:新型亲环素结合剂的鉴定》,《Journal of Molecular Biology(J. Mol. Biol.)》,第429卷,2017年



