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X-RAY STRUCTURE OF MPS1 IN COMPLEX WITH COMPOUND 16

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Protein Data Bank Japan2024-05-01 更新2026-03-21 收录
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X-RAY STRUCTURE OF MPS1 IN COMPLEX WITH COMPOUND 16 Descriptor: Dual specificity protein kinase TTK, [4-[[6-(3,5-dimethyl-4-oxidanyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]amino]phenyl]-morpholin-4-yl-methanone Authors: Marquardt, T, Holton, S.J, Schulze, V.K, Klar, U, Kosemund, D, Siemeister, G, Bader, B, Prechtl, S, Briem, H, Schirok, H, Bohlmann, R, Nguyen, D, Fernandez-Montalvan, A, Boemer, U, Eberspaecher, U, Brands, M, Nussbaum, F, Koppitz, M. Deposit date: 2019-12-06 Release date: 2020-05-13 Last modified: 2024-05-01 Method: X-RAY DIFFRACTION (2.6 Å) Cite: Treating Cancer by Spindle Assembly Checkpoint Abrogation: Discovery of Two Clinical Candidates, BAY 1161909 and BAY 1217389, Targeting MPS1 Kinase. J.Med.Chem., 63, 2020
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2019-12-06
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