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CryoEM structure of beta-2-adrenergic receptor in complex with GTP-bound Gs heterotrimer (transition intermediate #4 of 20)

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Protein Data Bank Japan2024-11-13 更新2026-05-23 收录
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CryoEM structure of beta-2-adrenergic receptor in complex with GTP-bound Gs heterotrimer (transition intermediate #4 of 20) Descriptor: (5R,6R)-6-(methylamino)-5,6,7,8-tetrahydronaphthalene-1,2,5-triol, Beta-2 adrenergic receptor, GUANOSINE-5'-TRIPHOSPHATE, ... Authors: Papasergi-Scott, M.M, Skiniotis, G. Deposit date: 2023-03-08 Release date: 2024-03-06 Last modified: 2024-11-13 Method: ELECTRON MICROSCOPY (3 Å) Cite: Time-resolved cryo-EM of G-protein activation by a GPCR. Nature, 629, 2024

结合有GTP的Gs异三聚体(GTP-bound Gs heterotrimer)与β2肾上腺素能受体(beta-2-adrenergic receptor)形成复合物的冷冻电镜(CryoEM)结构,对应20个过渡中间体中的第4号。描述项:(5R,6R)-6-(甲氨基)-5,6,7,8-四氢萘-1,2,5-三醇、β2肾上腺素能受体、鸟苷-5'-三磷酸(GUANOSINE-5'-TRIPHOSPHATE)…… 作者:帕帕塞尔吉-斯科特(Papasergi-Scott)M.M.、斯基尼奥蒂斯(Skiniotis)G. 存放日期:2023-03-08 发布日期:2024-03-06 最后修改日期:2024-11-13 方法:电子显微镜(ELECTRON MICROSCOPY),分辨率3 Å。引用文献:"Time-resolved cryo-EM of G-protein activation by a GPCR",《自然》(Nature),629卷,2024年。

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2023-03-08
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