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Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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Crystal Structure of PDE10A with Novel Keto-Benzimidazole Inhibitor Descriptor: 2-{4-[(6,7-difluoro-1H-benzimidazol-2-yl)amino]phenoxy}-N-methyl-3,4'-bipyridin-2'-amine, GLYCEROL, SULFATE ION, ... Authors: Chmait, S, Jordan, S. Deposit date: 2013-09-23 Release date: 2013-10-23 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.639 Å) Cite: Design, Optimization, and Biological Evaluation of Novel Keto-Benzimidazoles as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A). J.Med.Chem., 56, 2013
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2013-09-23
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