Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to ZS1-588
收藏Protein Data Bank Japan2023-10-18 更新2026-03-28 收录
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Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to ZS1-588 Descriptor: 1,2-ETHANEDIOL, 4-(6-{1-[(R)-S-methanesulfonimidoyl]cyclopropyl}-2-[(3R)-3-methylmorpholin-4-yl]pyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridine, DIMETHYL SULFOXIDE, ... Authors: Karim, M.R, Schonbrunn, E. Deposit date: 2021-12-04 Release date: 2022-01-19 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.89 Å) Cite: Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to ZS1-588 To Be Published
人源TAF1的串联溴结构域(bromodomain)BD1与BD2与ZS1-588结合的晶体结构
配体描述:1,2-乙二醇、4-(6-{1-[(R)-S-甲磺酰亚胺基]环丙基}-2-[(3R)-3-甲基吗啉-4-基]嘧啶-4-基)-1H-吡咯并[2,3-b]吡啶、二甲基亚砜等
作者:Karim M.R.、Schonbrunn E.
提交日期:2021-12-04
发布日期:2022-01-19
末次修改日期:2023-10-18
实验方法:X射线衍射(分辨率1.89埃)
引用:人源TAF1的串联溴结构域(BD1、BD2)与ZS1-588结合的晶体结构,待发表
创建时间:
2021-12-04



