Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus diazepam
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Human GABAA receptor alpha1-beta2-gamma2 subtype in complex with GABA plus diazepam Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 7-CHLORO-1-METHYL-5-PHENYL-1,3-DIHYDRO-2H-1,4-BENZODIAZEPIN-2-ONE, ... Authors: Kim, J.J, Gharpure, A, Teng, J, Zhuang, Y, Howard, R.J, Zhu, S, Noviello, C.M, Walsh, R.M, Lindahl, E, Hibbs, R.E. Deposit date: 2020-05-21 Release date: 2020-09-09 Last modified: 2024-11-20 Method: ELECTRON MICROSCOPY (2.92 Å) Cite: Shared structural mechanisms of general anaesthetics and benzodiazepines. Nature, 585, 2020
结合γ-氨基丁酸(GABA)与地西泮(diazepam)的人源γ-氨基丁酸A型受体(GABAA receptor)α1-β2-γ2亚型
描述符:2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖、2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖-(1→4)-2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖、7-氯-1-甲基-5-苯基-1,3-二氢-2H-1,4-苯并二氮杂䓬-2-酮……
作者:Kim, J.J.、Gharpure, A.、Teng, J.、Zhuang, Y.、Howard, R.J.、Zhu, S.、Noviello, C.M.、Walsh, R.M.、Lindahl, E.、Hibbs, R.E.
保藏日期:2020-05-21
发布日期:2020-09-09
最后修改日期:2024-11-20
实验方法:电子显微镜(分辨率2.92埃)
引用文献:《通用麻醉剂与苯二氮䓬类药物的共同结构机制》,《自然》(Nature),第585卷,2020年
创建时间:
2020-05-21



